Canakinumab

Anti-IL-1beta monoclonal antibody

Response rate
67.5% complete response
Onset
Days-weeks
Route
SC 150mg every 4-8 weeks
Line
2nd
IgM effect
Normalises SAA/CRP

Evidence summary

FDA and EMA approved for FMF. Longer dosing interval than anakinra (every 4-8 weeks vs daily). Reduced attacks from 8.3 to 1.56 per 24 weeks (P<0.001) in one cohort. Effective after colchicine and/or anakinra failure. Preferred by 72.2% of clinicians for colchicine-resistant FMF in multinational survey.

Molecular targets (1)

MoleculeRoleExpressionEvidence
IL-1βCentral effector cytokineElevatedestablished